Exercise 10
Key ... 110 pts
{A. Insight II on an SGI Computer}
{1. Logon to an SGI computer and activate Netscape Communicator}
{2. Activate Insight II}
{3. Insight II documentation}
Comments on Insight II documentation
??? [5 pts]
{B. The Insight II tutorial "Getting Started with Insight II"}
{1. Activate the Insight II tutorial "Getting Started with Insight II"}
{2. Do the Insight II tutorial}
{a. The "cheaters" way of doing the Tutorial}
{b. A "better" way of doing the Tutorial}
{c. The first Three Pages of Commands in the Tutorial: use of Lysozyme}
{d. Include comments in your Notebook}
Some comments on specific issues with
the tutorial ... [10 pts]
{e. Answer the Questions as you proceed through the Tutorial}
{C. Questions: }
1. What is Insight II and what does it do? [6
pts]
InsightII is a 3D graphical environment
for molecular modeling, best know for protein work, that runs
on Silicon Graphics (SGI) workstations. It creates, modifies,
naipulates, displays, and analyses molecular systems and related
data.
2. What are the modules in the Insight II package, and what
do each do? [6 pts]
Insight II has many modules; see URL http://www.accelrys.com/insight/
Also see the URL: http://www.accelrys.com/pdf/insight/i2_integrated_modeling_env.pdf
2 pts each
for any three, including something about their function or purpose:
Builder, Biopolymer, DelPhi, Solvation,
Discover, Discover_3, CHARMm, Docking, Ludi, Homology, Binding_site,
Ampac/Mopac, DMol, Turbomol, Zindo, QuanteMM
3. What are 4 additional applications in the MSI package, and
what does each do? [8 pts]
Many possibilities here also, see URL:
http://www.accelrys.com/
Some of these include: Quant and CNX
for protein x-ray crystallography, FELIX for NMR, Cerius@ for
protein simulation; GCG and MacVector for sequence analysis; SeqLab
and SeqWeb for graphical interfaces
4. How does one use the mouse to translate and rotate a protein
model? [3 pts]
To translate, use the middle button: the
model moves in the direction of mouse movement.
To rotate, press the right button; rotation
occurs in the direction of mouse movement
5. How are rotations in each of the three dimensions (about
x,y,z axes) correlated with motion of the mouse? [6
pts]
In ways that are strange to determine ....
two motions of the mouse for rotations about three axes ...
6. In what three different ways does one make choices using
the pulldown menus? [6 pts]
a) click on the choices in the pulldown
menu
b) click on a check box
c) type in a name in a given box ...
7. What is the comparable way of making choices using the command
line? [3 pts]
Type in the names of the commands on the
command line. Spaces occur between some and not others.
If a command is NOT chosen, use a minus sign in front of it.
8. What is the function of the Temperature Spectrum? [3 pts]
This shows the relative reactivity of each
type of amino acid residue.
9. What happends to the cylinders and ribbons when you rotate
the molecule? why is this? [6 pts]
They become stick characters from the solid,
blended characters, and are all of one color. This is to
save computation time during the redraw operations in the rotations.
10. How are hydrogen atoms represented in Insight II? [3 pts]
They are represented by horizontal-vertical
crosses ...
11. What is a subset of atoms and how are such used in Insight
II? [4 pts]
A subset of atoms is a group of atoms involved
in common structure or function. Insight II uses such from
graphical depiction of structure or function.
12. How is the subset called ACTIVE_SITE used in the tutorial?
[3 pts]
This is used as an example of a subset,
whose surface is solified, to show the surface of the lysozyme
active site.
13. What are the three numbers used to choose a "color"
in Insight II such as used in the color for the active_site atom
subset? [3 pts]
These show the relative mixtures of the
three primary colors (red, yellow, blue) used to give the chosen
color.
14. What "Molecular_Spec" was used in the "Create
Surface" operation for the Active Site, and why? [3 pts]
The Molecular_Spec is the "active_site"
subset of the Lysozyme residues, the subset of which one wishes
to create the surface graphic.
15. Why does the solid surface become a series of dots when
the molecule is rotated? [3 pts]
Same as Q.7 ... to save computation time
during the redraw opearations in the rotations.
16. What are the four steps in displaying the electrostatic
potential in color of the active site surface? Include the
purpose of each step in your answer. [8
pts]
The first 3 steps create, compute, and display
the grid using the Docking module. This grid, called ACTIVE_SITE_VGRD,
is the framework for the electrostatic potential. The first
step creates this grid; the second computes within the grid the
electrostatic potential values, the third displays these.
The fourth step converts the displayed values into color values
which then are displayed on the active_site surface.
17. Why are the colors of the surface then adjusted? [3 pts]
The contrast is initially low; the colors
are adjusted to fit a max and min that more closely fits the electrostatic
potential values, thereby permitting use of a wider color spectrum.
18. Comment on the logic of the steps in building small docking
molecules. [3 pts]
This is done excruciatingly slowly, step
by step, identifying each atom involved in forming each covalent
bond, with subsequent changes in angles and translation and rotation
relative to the protein, as needed for docking.
19. What is the substrate of Lysozyme, and how does the molecule
you constructed mimic this substrate? [6
pts]
Substrate is the peptidoglycan layer of
bacteria, a crosslinked molecule of amino acids and carbohydrate;
lysozyme cleaves linkages between glucose moities. The constructed
molecule contains a couple of monosaccharide residues joined in
the linkage cleaved hydrolytically by lysozyme.
20. Based on this substrate, why do you think tears from eyes
are a good source of lysozyme? [3 pts]
Lysozyme is found at high concentration
in tears to lyse bacteria that land on the surface of your eyes.
21. What does the energy minimization step in the Discover
module do? [6 pts]
This uses an iterative descent algorithm
to minimize the energy of the structure. In so doing, it
modifies angles slightly to yield a structure with energy equal
to that of the closest local minimum. Here we use 100 iterations
in this step.